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Jump to: 2014 | 2011 | 2010 | 2009 | 2008 | 2005 | 2004
Number of items: 12.

2014

Lu, Tiangong; Goh , Aik Wye; Yu, Mingfeng; Adams, Julian; Lam, Frankie; Teo, Theodosia; Li, Peng; Noll, Ben; Zhong, Longjin; Diab, Sarah; Chahrour, Osama; Hu, Anran; Abbas, Abdullahi Y,; Liu, Xiangrui; Huang, Shiliang; Sumby, Christopher J.; Milne, Robert; Midgley, Carol and Wang, Shudong (2014). Discovery of (E)-3-((styrylsulfonyl)methyl)pyridine and (E)-2-((styrylsulfonyl)methyl)pyridine derivatives as anticancer agents: synthesis, structure-activity relationships, and biological activities. Journal of Medicinal Chemistry, 57(6) pp. 2275–2291.

2011

Stachulski, Andrew V.; Pidathala, Chandrakala; Row, Eleanor C.; Sharma, Raman; Berry, Neil G.; Iqbal, Mazhar; Bentley, Joanne; Allman, Sarah A.; Edwards, Geoffrey; Helm, Alison; Hellier, Jennifer; Korba, Brent E.; Semple, J. Edward and Rossignol, Jean-Francois (2011). Thiazolides as novel antiviral agents. 1. Inhibition of hepatitis B virus replication. Journal of Medicinal Chemistry, 54(12) pp. 4119–4132.

Stachulski, Andrew V.; Pidathala, Chandrakala; Row, Eleanor C.; Sharma, Raman; Berry, Neil G.; Lawrenson, Alexandre S.; Moores, Shelley L.; Iqbal, Mazhar; Bentley, Joanne; Allman, Sarah A.; Edwards, Geoffrey; Helm, Alison; Hellier, Jennifer; Korba, Brent E.; Semple, J. Edward and Rossignol, Jean-Francois (2011). Thiazolides as novel antiviral agents. 2. Inhibition of Hepatitis C virus replication. Journal of Medicinal Chemistry, 54(24) pp. 8670–8680.

2010

Mulchande, Jalmira; Oliveira, Rudi; Carrasco, Marta; Gouveia, Luís; Guedes, Rita C.; Iley, Jim and Moreira, Rui (2010). 4-Oxo-β-lactams (Azetidine-2,4-diones) Are Potent and Selective Inhibitors of Human Leukocyte Elastase. Journal of Medicinal Chemistry, 53(1) pp. 241–253.

Wang, Shudong; Midgley, Carol A.; Scaërou, Frederic; Grabarek, Joanna B.; Griffiths, Gary; Jackson, Wayne; Kontopidis, George; McClue, Steven J.; McInnes, Campbell; Meades, Christopher; Mezna, Mokdad; Plater, Andy; Stuart, Iain; Thomas, Mark P.; Wood, Gavin; Clarke, Rosemary G.; Blake, David G.; Zheleva, Daniella I.; Lane, David P.; Jackson, Robert C.; Glover, David M. and Fischer, Peter M. (2010). Discovery of N-Phenyl-4-(thiazol-5-yl)pyrimidin-2-amine Aurora Kinase Inhibitors. Journal of Medicinal Chemistry, 53(11) pp. 4367–4378. restricted access item, not available for direct downloadfile

2009

Perry, M. J.; Mendes, E.; Simplício, A. L.; Coelho, A.; Iley, J.; Moreira, R. and Francisco, A. P. (2009). Dopamine- and tyramine-based derivatives of triazenes. Activation by tyrosinase and implications for prodrug design. European Journal of Medicinal Chemistry, 44(8) pp. 3228–3234. file

Perry, Maria de Jesus; Carvalho, Emília; Rosa, Eduarda and Iley, Jim (2009). Towards an efficient prodrug of the alkylating metabolite monomethyltriazene: Synthesis and stability of N-acylamino acid derivatives of triazenes. European Journal of Medicinal Chemistry, 44(3) pp. 1049–1056. file

2008

Cheng, Mai-Kim; Modi, Chetna; Cookson, Jennifer C.; Hutchinson, Ian; Heald, Robert A.; McCarroll, Andrew J.; Missailidis, Sotiris; Tanious, Farial; Wilson, W. David; Mergny, Jean-Louis; Laughton, Charles A. and Stevens, Malcolm F. G. (2008). Antitumor Polycyclic Acridines. 20. Search for DNA Quadruplex Binding Selectivity in a Series of 8,13-Dimethylquino[4,3,2-kl]acridinium Salts: Telomere-Targeted Agents. Journal of Medicinal Chemistry, 51(4) pp. 963–975.

Mulchande, J.; Guedes, R. C.; Tsang, W.-Y.; Page, M. I.; Moreira, R. and Iley, J. (2008). Azetidine-2,4-diones (4-oxo-beta-lactams) as scaffolds for designing elastase inhibitors. Journal of Medicinal Chemistry, 51(6) pp. 1783–1790.

2005

Araújo, Maria Joao; Bom, Joana; Capela, Rita; Casimiro, Catarina; Chambel, Paula; Gomes, Paula; Iley, Jim; Lopes, Francisca; Morais, Jose; Moreira, Rui; de Oliveira, Eliandre; do Rosário, Virgilio and Vale, Nuno (2005). Imidazolidin-4-one derivatives of primaquine as novel transmission-blocking antimalarials. Journal of Medicinal Chemistry, 48 pp. 888–892.

Moreira, Rui; Santana, Ana Bela; Iley, Jim; Neres, Joao; Douglas, Kenneth T.; Horton, Peter N. and Hursthouse, Michael B. (2005). Design, Synthesis, and Enzymatic Evaluation of N1-Acyloxyalkyl- and N1-Oxazolidin-2,4-dion-5-yl-Substituted beta-lactams as Novel Inhibitors of Human Leukocyte Elastase. Journal of Medicinal Chemistry, 48(15) pp. 4861–4870.

2004

Wang, Shudong; Meades, Christopher; Wood, Gavin; Osnowski, Andrew; Anderson, Sian; Yuill, Rhoda; Thomas, Mark; Mezna, Mokdad; Jackson, Wayne; Midgley, Carol; Griffiths, Gary; Fleming, Ian; Green, Simon; McNae, Ian; Wu, Su-Ying; McInnes, Campbell; Zheleva, Daniella; Walkinshaw, Malcolm D. and Fischer, Peter M. (2004). 2-Anilino-4-(thiazol-5-yl)pyrimidine CDK Inhibitors: Synthesis, SAR Analysis, X-ray Crystallography, and Biological Activity. Journal of Medicinal Chemistry, 47(7) pp. 1662–1675.

This list was generated on Thu Oct 23 23:51:57 2014 BST.

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